5MRD | pdb_00005mrd

Human PDK1-PKCiota Kinase Chimera in Complex with Allosteric Compound PS267 Bound to the PIF-Pocket

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RCSB PDB Mol* Viewer 2.11.2 [1/27/2025, 4:56:27 PM]
Sequence of
     ​A​​M​​D​​G​​T​​A​​A​​E​​P​​R​     ​P​​G​​A​​G​​S​​L​​Q​​H​​A​​Q​     ​P​​P​​P​​Q​​P​​R​​S​​K​​R​​P​80   ​E​​D​​F​​K​​F​​G​​K​​I​​L​​G​90   ​E​​G​​S​​F​​S​​T​​V​​V​​L​​A​100  ​R​​E​​L​​A​​T​​S​​R​​E​​Y​​A​110  ​I​​K​​I​​V​​E​​K​​R​​H​​V​​N​120  ​K​​E​​N​​K​​I​​P​​Y​​V​​Q​​R​130  ​E​​K​​D​​V​​M​​S​​R​​L​​D​​H​140  ​P​​F​​F​​V​​K​​L​​Y​​F​​C​​F​150  ​Q​​D​​D​​E​​K​​L​​Y​​F​​G​​L​160  ​S​​Y​​A​​K​​N​​G​​E​​L​​L​​K​170  ​Y​​I​​R​​K​​I​​G​​S​​F​​D​​E​180  ​T​​C​​T​​R​​F​​Y​​T​​A​​E​​I​190  ​V​​S​​A​​L​​E​​Y​​L​​H​​G​​K​200  ​G​​I​​I​​H​​R​​D​​L​​K​​P​​E​210  ​N​​I​​L​​L​​N​​E​​D​​M​​H​​I​220  ​Q​​I​​T​​D​​F​​G​​T​​A​​K​​V​230  ​L​​S​​P​​E​​S​​K​​Q​​A​​R​​A​240  ​N​​SEP​​F​​V​​G​​T​​A​​Q​​Y​​V​250  ​S​​P​​E​​L​​L​​T​​E​​K​​S​​A​260  ​C​​K​​S​​S​​D​​L​​W​​A​​L​​G​270  ​C​​I​​I​​Y​​Q​​L​​V​​A​​G​​L​280  ​P​​P​​F​​R​​A​​G​​N​​E​​G​​L​290  ​I​​F​​A​​K​​I​​I​​K​​L​​E​​Y​300  ​D​​F​​P​​E​​K​​F​​F​​P​​K​​A​310  ​R​​D​​L​​V​​E​​K​​L​​L​​V​​L​320  ​D​​A​​T​​K​​R​​L​​G​​C​​E​​E​330  ​M​​E​​G​​Y​​G​​P​​L​​K​​A​​H​340  ​P​​F​​F​​E​​S​​V​​T​​W​​E​​N​350  ​L​​H​​Q​​Q​​T​​P​​P​​K​​L​​T​
Type
Asm Id
Dynamic Bonds

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