6NFA | pdb_00006nfa

Vav1 inhibited by an allosteric inhibitor: Vav1 inhibitors block GEF activity

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RCSB PDB Mol* Viewer 2.11.2 [1/27/2025, 4:56:27 PM]
Sequence of
     ​M​​G​​K​​H​​H​​H​​H​​H​​H​​E​     ​N​​L​​Y​​F​​Q​​G​​D​​E​​I​​Y​175  ​E​​D​​L​​M​​R​​S​​E​​P​​V​​S​     ​M​​P​​P​​K​​M​​T​​E​​Y​​D​​K​195  ​R​​C​​C​​C​​L​​R​​E​​I​​Q​​Q​205  ​T​​E​​E​​K​​Y​​T​​D​​T​​L​​G​215  ​S​​I​​Q​​Q​​H​​F​​L​​K​​P​​L​225  ​Q​​R​​F​​L​​K​​P​​Q​​D​​I​​E​235  ​I​​I​​F​​I​​N​​I​​E​​D​​L​​L​245  ​R​​V​​H​​T​​H​​F​​L​​K​​E​​M​255  ​K​​E​​A​​L​​G​​T​​P​​G​​A​​A​265  ​N​​L​​Y​​Q​​V​​F​​I​​K​​Y​​K​275  ​E​​R​​F​​L​​V​​Y​​G​​R​​Y​​C​285  ​S​​Q​​V​​E​​S​​A​​S​​K​​H​​L​295  ​D​​R​​V​​A​​A​​A​​R​​E​​D​​V​305  ​Q​​M​​K​​L​​E​​E​​C​​S​​Q​​R​315  ​A​​N​​N​​G​​R​​F​​T​​L​​R​​D​325  ​L​​L​​M​​V​​P​​M​​Q​​R​​V​​L​335  ​K​​Y​​H​​L​​L​​L​​Q​​E​​L​​V​345  ​K​​H​​T​​Q​​E​​A​​M​​E​​K​​E​355  ​N​​L​​R​​L​​A​​L​​D​​A​​M​​R​365  ​D​​L​​A​​Q​​C​​V​​N​​E​​V​​K​375  ​R​​D​​N​​E​​T​​L​​R​​Q​​I​​T​385  ​N​​F​​Q​​L​​S​​I​​E​​N​​L​​D​395  ​Q​​S​​L​​A​​H​​Y​​G​​R​​P​​K​405  ​I​​D​​G​​E​​L​​K​​I​​T​​S​​V​415  ​E​​R​​R​​S​​K​​M​​D​​R​​Y​​A​425  ​F​​L​​L​​D​​K​​A​​L​​L​​I​​C​435  ​K​​R​​R​​G​​D​​S​​Y​​D​​L​​K​445  ​D​​F​​V​​N​​L​​H​​S​​F​​Q​​V​455  ​R​​D​​D​​S​​S​​G​​D​​R​​D​​N​465  ​K​​K​​W​​S​​H​​M​​F​​L​​L​​I​475  ​E​​D​​Q​​G​​A​​Q​​G​​Y​​E​​L​485  ​F​​F​​K​​T​​R​​E​​L​​K​​K​​K​495  ​W​​M​​E​​Q​​F​​E​​M​​A​​I​​S​505  ​N​​I​​Y​​P​​E​​N​​A​​T​​A​​N​515  ​G​​H​​D​​F​​Q​​M​​F​​S​​F​​E​525  ​E​​T​​T​​S​​C​​K​​A​​C​​Q​​M​535  ​L​​L​​R​​G​​T​​F​​Y​​Q​​G​​Y​545  ​R​​C​​H​​R​​C​​R​​A​​S​​A​​H​555  ​K​​E​​C​​L​​G​​R​​V​​P​​P​​C​565  ​G​​R​​H​​G​​Q​​D​​F​​P​​G​​T​     ​M​
Type
Asm Id
Dynamic Bonds

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