3SDG | pdb_00003sdg

Ethionamide Boosters Part 2: Combining Bioisosteric Replacement and Structure-Based Drug Design to Solve Pharmacokinetic Issues in a Series of Potent 1,2,4-Oxadiazole EthR Inhibitors.

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CHAIN
A
Transcription initiation factor TFIID subunit 1 - Homo sapiens
 Explore Sequence Annotations in 3D
020406080100120140
CHAIN A
GSPLLDDDDQVAFSFILDNIVTQKMMAVPDSWPFHHPVNKKFVPDYYKVIVNPMDLETIRKNISKHKYQSRESFLDDVNLILANSVKYNGPESQYTKTAQEIVNVCYQTLTEYDEHLTQLEKDICTAKEAALEEAELESLDPMT
UNIPROT P21675
PLLDDDDQVAFSFILDNIVTQKMMAVPDSWPFHHPVNKKFVPDYYKVIVNPMDLETIRKNISKHKYQSRESFLDDVNLILANSVKYNGPESQYTKTAQEIVNVCYQTLTEYDEHLTQLEKDICTAKEAALEEAELESLDPMT
SECONDARY STRUCTURE
UNMODELED
EDS ATOMS
OCC WT AVG B
AVERAGE OCCUPANCY
ATOMIC CLASHES
ANGLE OUTLIERS
BOND OUTLIERS
RSRZ
RSR
RSCC
BURIED RESIDUES
ARTIFACT
HYDROPATHY
DISORDER
DISORDERED BINDING
PFAM
CATH
SCOP
ECOD
MOLECULE PROCESSING
DOMAIN
REGION
COMPOSITIONAL BIAS
SEQUENCE SPLICING